ICI-118551

Catalog No.: A15878

β2 adrenergic receptor antagonist

ICI-118551

ICI-118551 Chemical Structure

CAS NO. 1217094-53-5

ICI-118551 is a selective beta2 adrenergic receptor (adrenoreceptor) antagonist.

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10 mg
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25 mg
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50 mg
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  • Moon Jain, .et al. Involvement of angiotensin II and beta-adrenergic receptors in the regulation of autophagy in human endothelial EA.hy926 cell line, Tropical Journal of Pharmaceutical Research, 2020, Vol. 19 No. 4

Biological Activity

ICI-118551 is a selective beta2 adrenergic receptor (adrenoreceptor) antagonist.
Targets
β2-adrenergic receptor β1-adrenergic receptor β3-adrenoceptor
0.7nM(Ki)49.5nM(Ki)611nM(Ki)
In vitro DMSO 59 mg/mL (187.98 mM)
Water 20 mg/mL (63.71 mM)
Ethanol 59 mg/mL (187.98 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 31.86 mL 159.31 mL 318.61 mL
0.5 mM 6.37 mL 31.86 mL 63.72 mL
1 mM 3.19 mL 15.93 mL 31.86 mL
5 mM 0.64 mL 3.19 mL 6.37 mL

*The above data is based on the productmolecular weight 313.86. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15878
Actions Antagonist
CAS No. 1217094-53-5
Formula C17H27NO2.HCl
M. Wt 313.86
Solubility DMSO
Purity >98%
Synonyms ICI118551, ICI 118551
SMILES CC1=C(CCC2)C2=C(OC[[email protected]](O)[[email protected]@H](C)NC(C)C)C=C1.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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