Keap1-Nrf2-IN-5

Name: Keap1-Nrf2-IN-5
Brand: Adooq Bioscience
SKU: A79529
Rating: 5 (288 reviews)

Catalog No.: A79529

Keap1-Nrf2 PPI Inhibitor

Keap1-Nrf2-IN-5 is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), with an IC50 of 4.1 µM and a Kd of 3.7 µM. This compound enhances Nrf2 activity, promoting the expression of antioxidant and cytoprotective genes. It serves as a valuable tool for research into oxidative stress, neuroprotection, and cancer therapeutics.

Skip to the end of the images gallery

Keap1-Nrf2-IN-5 2696272-70-3 Keap1-Nrf2 PPI Inhibitor

Skip to the beginning of the images gallery

Grouped product items
Size	Price	Stock
25mg	$1,800.00	In stock
50mg	$2,285.00	In stock
100mg	$2,815.00	In stock
Bulk Size	Bulk Discount

Bulk Inquiry

Notify me when the price drops

Free Delivery on orders over $500

Research use only. We do not sell to patients.

Data Sheet SDS

Loading distributor info...

Adooq Products cited in reputable paper

Biological Activity

Description	Keap1-Nrf2-IN-5 is a potent inhibitor of the Keap1-Nrf2 protein-protein interaction (PPI), with an IC50 of 4.1 µM and a Kd of 3.7 µM. This compound enhances Nrf2 activity, promoting the expression of antioxidant and cytoprotective genes. It serves as a valuable tool for research into oxidative stress, neuroprotection, and cancer therapeutics.

Product Information

Catalog Num	A79529
Formula	C23H30N4O6S
Molecular Weight	490.57
CAS Number	2696272-70-3
SMILES	O=C([C@H](NC([C@H](NC([C@H]1N(C(C)=O)CCC1)=O)CO2)=O)CSCC3=CC=CC=C3C2=O)N(C)C

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂