Ketoconazole

Catalog No.: A10498

P450 inhibitor

Ketoconazole

Ketoconazole Chemical Structure

CAS NO. 65277-42-1

As an antifungal, ketoconazole is structurally similar to imidazole, and interferes with the fungal synthesis of ergosterol, a constituent of fungal cell membranes, as well as certain enzymes.

Availability: In stock

Package Price Qty
100 mg

Regular Price: $50.00

Special Price $40.00

200 mg

Regular Price: $85.00

Special Price $68.00

500 mg

Regular Price: $150.00

Special Price $120.00

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

As an antifungal, ketoconazole is structurally similar to imidazole, and interferes with the fungal synthesis of ergosterol, a constituent of fungal cell membranes, as well as certain enzymes.
Targets
Cyclosporine oxidase Testosterone 6 beta-hydroxylase
0.19 mM0.22 mM
In vitro (25°C) DMSO Warmed: 5 mg/mL (9.4 mM)
Water Insoluble
Ethanol 7 mg/mL
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.82 mL 94.09 mL 188.18 mL
0.5 mM 3.76 mL 18.82 mL 37.64 mL
1 mM 1.88 mL 9.41 mL 18.82 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 531.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10498
Actions Inhibitor
CAS No. 65277-42-1
Formula C26H28Cl2N4O4
M. Wt 531.4
Purity >98%
Synonyms Nizoral, Extina, Xolegel, Kuric
SMILES CC(=O)N1CCN(CC1)C2=CC=C(C=C2)OC[[email protected]]3CO[[email protected]](O3)(CN4C=CN=C4)C5=C(C=C(C=C5)Cl)Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Ketoconazole | Ketoconazole Supplier | purchase | cost | manufacturer | order | distributor | buy 65277-42-1| 65277-42-1 Supplier | purchase 65277-42-1 | 65277-42-1 cost | 65277-42-1 manufacturer | order 65277-42-1 | 65277-42-1 distributor
Rewards