Ketoconazole

Catalog No.: A10498

P450 inhibitor

Ketoconazole

Ketoconazole Chemical Structure

CAS NO. 65277-42-1

As an antifungal, ketoconazole is structurally similar to imidazole, and interferes with the fungal synthesis of ergosterol, a constituent of fungal cell membranes, as well as certain enzymes.

Availability: In stock

Package Price Qty
100 mg

Regular Price: $50.00

Special Price $45.00

200 mg

Regular Price: $85.00

Special Price $76.50

500 mg

Regular Price: $150.00

Special Price $135.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

As an antifungal, ketoconazole is structurally similar to imidazole, and interferes with the fungal synthesis of ergosterol, a constituent of fungal cell membranes, as well as certain enzymes.
Targets
Cyclosporine oxidase Testosterone 6 beta-hydroxylase
0.19 mM0.22 mM
In vitro (25°C) DMSO 3 mg/mL (5.64 mM)
Water <1 mg/mL (<1 mM)
Ethanol 7 mg/mL (13.17 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.82 mL 94.09 mL 188.18 mL
0.5 mM 3.76 mL 18.82 mL 37.64 mL
1 mM 1.88 mL 9.41 mL 18.82 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 531.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10498
Actions Inhibitor
M. Wt 531.4
Formula C26H28Cl2N4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 65277-42-1
Synonyms Nizoral, Extina, Xolegel, Kuric
SMILES CC(=O)N1CCN(CC1)C2=CC=C(C=C2)OC[[email protected]]3CO[[email protected]](O3)(CN4C=CN=C4)C5=C(C=C(C=C5)Cl)Cl

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