Lerociclib dihydrochloride

Catalog No.: A21577

CDK4/CDK6 inhibitor

Lerociclib dihydrochloride

Lerociclib dihydrochloride Chemical Structure

CAS NO. 2097938-59-3

Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively.

Availability: In stock

Package Price Qty
5 mg
$495.00
10 mg
$853.00
50 mg
$2,530.00
100 mg
$5,060.00
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Biological Activity

Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.26 mL 91.32 mL 182.64 mL
0.5 mM 3.65 mL 18.26 mL 36.53 mL
1 mM 1.83 mL 9.13 mL 18.26 mL
5 mM 0.37 mL 1.83 mL 3.65 mL

*The above data is based on the productmolecular weight 547.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21577
Actions Inhibitor
M. Wt 547.52
Formula C26H36Cl2N8O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2097938-59-3
Synonyms G1T38 dihydrochloride, G1T 38, G1T-38
SMILES O=C1NCC2(N3C1=CC4=CN=C(NC5=NC=C(N6CCN(C(C)C)CC6)C=C5)N=C43)CCCCC2.[H]Cl.[H]Cl

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