LJH685

Catalog No.: A14372

pan-RSK inhibitor

LJH685

LJH685 Chemical Structure

CAS NO. 1627710-50-2

LJH685 is a potent , specific and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50 of 4 to 13 nM.

Availability: In stock

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5 mg

Regular Price: $90.00

Special Price $72.00

10 mg

Regular Price: $150.00

Special Price $120.00

25 mg

Regular Price: $300.00

Special Price $240.00

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Biological Activity

LJH685 is a potent , specific and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50 of 4 to 13 nM.
Targets
RSK3 RSK2 RSK1
4 nM5 nM6 nM
In vitro DMSO 66 mg/mL (173.03 mM)
Water Insoluble
Ethanol 17 mg/mL (44.57 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.22 mL 131.09 mL 262.18 mL
0.5 mM 5.24 mL 26.22 mL 52.44 mL
1 mM 2.62 mL 13.11 mL 26.22 mL
5 mM 0.52 mL 2.62 mL 5.24 mL

*The above data is based on the productmolecular weight 381.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14372
Actions Inhibitor
CAS No. 1627710-50-2
Formula C22H21F2N3O
M. Wt 381.42
Purity >98%
Synonyms LJH 685, LJH-685
SMILES CN(CC1)CCN1C(C=C2)=CC=C2C3=CC=NC=C3C4=CC(F)=C(O)C(F)=C4
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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