Customer Appreciation Sale.
15% off with promo code "APPRECIATION2023" on check out or purchase order
Biological Activity
LJH685 is a potent , specific and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50 of 4 to 13 nM.
Targets
RSK3 | RSK2 | RSK1 | ||
4 nM | 5 nM | 6 nM |
In vitro | DMSO | 66 mg/mL (173.03 mM) | |
Water | Insoluble | ||
Ethanol | 17 mg/mL (44.57 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 26.22 mL | 131.09 mL | 262.18 mL |
0.5 mM | 5.24 mL | 26.22 mL | 52.44 mL |
1 mM | 2.62 mL | 13.11 mL | 26.22 mL |
5 mM | 0.52 mL | 2.62 mL | 5.24 mL |
*The above data is based on the productmolecular weight 381.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A14372 |
---|---|
Actions | Inhibitor |
CAS No. | 1627710-50-2 |
Formula | C22H21F2N3O |
M. Wt | 381.42 |
Purity | >98% |
Synonyms | LJH 685, LJH-685 |
SMILES | CN(CC1)CCN1C(C=C2)=CC=C2C3=CC=NC=C3C4=CC(F)=C(O)C(F)=C4 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy LJH685 | LJH685 Supplier | purchase | cost | manufacturer | order | distributor | buy 1627710-50-2| 1627710-50-2 Supplier | purchase 1627710-50-2 | 1627710-50-2 cost | 1627710-50-2 manufacturer | order 1627710-50-2 | 1627710-50-2 distributor