Lomitapide mesylate

Catalog No.: A16600

MTP inhibitor

Lomitapide mesylate

Lomitapide mesylate Chemical Structure

CAS NO. 202914-84-9

Lomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.

Availability: In stock

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1 mg

Regular Price: $320.00

Special Price $256.00

5 mg

Regular Price: $960.00

Special Price $768.00

10 mg

Regular Price: $1,600.00

Special Price $1,280.00

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Biological Activity

Lomitapide mesylate(AEGR-733; BMS-201038) is an inhibitor of microsomal triglyceride-transfer protein (MTP) wtih in vitro IC50 of 8 nM.
In vitro DMSO 91 mg/mL (115.21 mM)
Water Insoluble
Ethanol 91 mg/mL (115.21 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.66 mL 63.3 mL 126.61 mL
0.5 mM 2.53 mL 12.66 mL 25.32 mL
1 mM 1.27 mL 6.33 mL 12.66 mL
5 mM 0.25 mL 1.27 mL 2.53 mL

*The above data is based on the productmolecular weight 789.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16600
Actions Inhibitor
CAS No. 202914-84-9
Formula C40H41F6N3O5S
M. Wt 789.83
Purity >98%
Synonyms AEGR-733 mesylate, AEGR733, AEGR 733; BMS-201038 mesylate, BMS 201038, BMS201038
SMILES O=C(C1(CCCCN2CCC(NC(C3=CC=CC=C3C4=CC=C(C(F)(F)F)C=C4)=O)CC2)C5=C(C6=C1C=CC=C6)C=CC=C5)NCC(F)(F)F.O=S(C)(O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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