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LY3214996 is a selective and novel ERK1/2 inhibitor with IC50 of 5 nM for both enzymes in biochemical assays. It potently inhibits cellular phospho-RSK1 in BRAF and RAS mutant cancer cell lines.
| In vitro | DMSO | 24 mg/mL (52.91 mM) | |
| Water | Insoluble | ||
| Ethanol | 14 mg/mL (30.86 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 22.05 mL | 110.24 mL | 220.48 mL |
| 0.5 mM | 4.41 mL | 22.05 mL | 44.1 mL |
| 1 mM | 2.2 mL | 11.02 mL | 22.05 mL |
| 5 mM | 0.44 mL | 2.2 mL | 4.41 mL |
*The above data is based on the productmolecular weight 453.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A16843 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1951483-29-6 |
| Formula | C22H27N7O2S |
| M. Wt | 453.56 |
| Purity | >98% |
| Synonyms | LY 3214996, LY-3214996 |
| SMILES | CC(N(CCN1CCOCC1)C2=O)(C)C3=C2C=C(S3)C4=CC=NC(NC5=CC=NN5C)=N4 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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