MA-2029 is a selective, orally active antagonist of the motilin receptor, exhibiting an IC50 of 4.9 nM. It demonstrates high selectivity for the motilin receptor compared to a variety of other receptors and ion channels. This compound is particularly relevant for research into gastrointestinal disorders linked to impaired gastrointestinal motility, providing a valuable tool for studying motility-related pathophysiology and potential therapeutic interventions.
MA-2029 is a selective, orally active antagonist of the motilin receptor, exhibiting an IC50 of 4.9 nM. It demonstrates high selectivity for the motilin receptor compared to a variety of other receptors and ion channels. This compound is particularly relevant for research into gastrointestinal disorders linked to impaired gastrointestinal motility, providing a valuable tool for studying motility-related pathophysiology and potential therapeutic interventions.
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