MK-1064

Catalog No.: A16360

OX2 Antagonist

MK-1064

MK-1064 Chemical Structure

CAS NO. 1207253-08-4

MK-1064 is a potent, selective and orally active Orexin OX2 Receptor Antagonist for potential treatment of insomnia.

Availability: In stock

Package Price Qty
1 mg
$80.00
2 mg
$140.00
5 mg
$195.00
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Biological Activity

MK-1064 is a potent, selective and orally active Orexin OX2 Receptor Antagonist for potential treatment of insomnia.
In vitro DMSO 87 mg/mL (188.35 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.65 mL 108.25 mL 216.49 mL
0.5 mM 4.33 mL 21.65 mL 43.3 mL
1 mM 2.16 mL 10.82 mL 21.65 mL
5 mM 0.43 mL 2.16 mL 4.33 mL

*The above data is based on the productmolecular weight 461.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16360
Actions Antagonist
CAS No. 1207253-08-4
Formula C24H20ClN5O3
M. Wt 461.91
Purity >98%
Synonyms MK1064, MK 1064
SMILES O=C(C1=CC(C2=CC(Cl)=CN=C2)=CN=C1C3=NC=CC=C3)NCC4=NC(OC)=C(OC)C=C4
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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