MK-3102

Catalog No.: A13310

DPP-4 inhibitor

MK-3102

MK-3102 Chemical Structure

CAS NO. 1226781-44-7

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).

Availability: In stock

Package Price Qty
5 mg
$160.00
10 mg
$240.00
25 mg
$480.00
50 mg
$640.00
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Biological Activity

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.1 mL 125.49 mL 250.99 mL
0.5 mM 5.02 mL 25.1 mL 50.2 mL
1 mM 2.51 mL 12.55 mL 25.1 mL
5 mM 0.5 mL 2.51 mL 5.02 mL

*The above data is based on the productmolecular weight 398.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13310
Actions Inhibitor
M. Wt 398.43
Formula C17H20F2N4O3S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1226781-44-7
SMILES CS(=O)(=O)N1C=C2CN(CC2=N1)[[email protected]@H]3C[[email protected]@H]([[email protected]](OC3)C4=C(C=CC(=C4)F)F)N

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