Total item
Cart Subtotal
$0.00 Biological Activity
Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 25.1 mL | 125.49 mL | 250.99 mL |
| 0.5 mM | 5.02 mL | 25.1 mL | 50.2 mL |
| 1 mM | 2.51 mL | 12.55 mL | 25.1 mL |
| 5 mM | 0.5 mL | 2.51 mL | 5.02 mL |
*The above data is based on the productmolecular weight 398.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13310 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 398.43 |
| Formula | C17H20F2N4O3S |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1226781-44-7 |
| SMILES | CS(=O)(=O)N1C=C2CN(CC2=N1)[[email protected]@H]3C[[email protected]@H]([[email protected]](OC3)C4=C(C=CC(=C4)F)F)N |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy MK-3102 | MK-3102 Supplier | purchase MK-3102 | MK-3102 cost | MK-3102 manufacturer | order MK-3102 | MK-3102 distributor | buy 1226781-44-7| 1226781-44-7 Supplier | purchase 1226781-44-7 | 1226781-44-7 cost | 1226781-44-7 manufacturer | order 1226781-44-7 | 1226781-44-7 distributor
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: [email protected]
Not your Region? View all Distributors
Adooq Quality Guarantee
We promise all products perform as described.