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MK-3102

Catalog No.: A13310

DPP-4 inhibitor

MK-3102

MK-3102 Chemical Structure

CAS NO. 1226781-44-7

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $81.00

Special Price $64.80

10 mg

Regular Price: $138.00

Special Price $110.40

25 mg

Regular Price: $243.00

Special Price $194.40

50 mg

Regular Price: $405.00

Special Price $324.00

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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Omarigliptin (MK-3102) is a competitive, reversible inhibitor of DPP-4 (IC50 = 1.6 nM, Ki = 0.8 nM). It is highly selective over all proteases tested (IC50 > 67 μM), including QPP, FAP, PEP, DPP8, and DPP9 and has weak ion channel activity (IC50 > 30 μM at IKr, Caγ1.2, and Naγ1.5).
In vitro DMSO 77 mg/mL (193.25 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.1 mL 125.49 mL 250.99 mL
0.5 mM 5.02 mL 25.1 mL 50.2 mL
1 mM 2.51 mL 12.55 mL 25.1 mL
5 mM 0.5 mL 2.51 mL 5.02 mL

*The above data is based on the productmolecular weight 398.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13310
Actions Inhibitor
CAS No. 1226781-44-7
Formula C17H20F2N4O3S
M. Wt 398.43
Purity >98%
SMILES CS(=O)(=O)N1C=C2CN(CC2=N1)[[email protected]@H]3C[[email protected]@H]([[email protected]](OC3)C4=C(C=CC(=C4)F)F)N
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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