MM-102 TFA

Catalog No.: A21941

WDR5/MLL interaction inhibitor

MM-102 TFA

MM-102 TFA Chemical Structure

CAS NO. 1883545-52-5

MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.

Availability: In stock

Package Price Qty
2 mg

Regular Price: $54.00

Special Price $43.20

5 mg

Regular Price: $108.00

Special Price $86.40

10 mg

Regular Price: $210.00

Special Price $168.00

50 mg

Regular Price: $618.00

Special Price $494.40

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.76 mL 63.79 mL 127.58 mL
0.5 mM 2.55 mL 12.76 mL 25.52 mL
1 mM 1.28 mL 6.38 mL 12.76 mL
5 mM 0.26 mL 1.28 mL 2.55 mL

*The above data is based on the productmolecular weight 783.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21941
Actions Inhibitor
CAS No. 1883545-52-5
Formula C37H50F5N7O6
M. Wt 783.83
Purity >98%
Synonyms HMTase Inhibitor IX TFA, MM102, MM 102
SMILES O=C(C1(NC([[email protected]@H](NC(C(NC(C(C)C)=O)(CC)CC)=O)CCCNC(N)=N)=O)CCCC1)NC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3.FC(F)(F)C(O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy MM-102 TFA | MM-102 TFA Supplier | purchase | cost | manufacturer | order | distributor | buy 1883545-52-5| 1883545-52-5 Supplier | purchase 1883545-52-5 | 1883545-52-5 cost | 1883545-52-5 manufacturer | order 1883545-52-5 | 1883545-52-5 distributor
Rewards