MOR agonist-4

Catalog No.: A62434
KOR Agonist
MOR agonist-4 is a G protein signaling-biased agonist of the Kappa opioid receptor (KOR) with an EC50 value of 11 nM. This compound features an electron-withdrawing CF3 group and exhibits a bias factor of 38 based on triazole structure. It is primarily utilized in research related to pruritus and pain relief, facilitating the study of analgesic pathways and mechanisms.
Grouped product items
Size Price Stock Qty
5mg
$350.00
In stock
10mg
$650.00
In stock
50mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Nature Volume 622 Issue 7982 (2023)
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Nature volume 551, pages639-643 (2017)
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Biological Activity
DescriptionMOR agonist-4 is a G protein signaling-biased agonist of the Kappa opioid receptor (KOR) with an EC50 value of 11 nM. This compound features an electron-withdrawing CF3 group and exhibits a bias factor of 38 based on triazole structure. It is primarily utilized in research related to pruritus and pain relief, facilitating the study of analgesic pathways and mechanisms.
Product Information
Catalog NumA62434
FormulaC22H19F3N4S
Molecular Weight428.47
CAS Number3050669-97-8
SMILESCC(C=C1)=C(C(F)(F)F)C=C1CCC(N2CC3=CC=CS3)=NN=C2C4=CC=CC=N4
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