MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.
MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.
Targets
Target
Value
Product Information
Catalog Num
A13236
Formula
C14H11N.HCl
Molecular Weight
229.7
CAS Number
219911-35-0
SMILES
CC1=CC=CC(=N1)C#CC2=CC=CC=C2.Cl
Synonyms
MPEP hydrochloride
Storage
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
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