MPEP HCl

Catalog No.: A13236

mGlu5 receptor antagonist

MPEP HCl

MPEP HCl Chemical Structure

CAS NO. 219911-35-0

MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.

Availability: In stock

Package Price Qty
25 mg
$120.00
50 mg
$200.00
100 mg
$350.00
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Biological Activity

MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 43.54 mL 217.68 mL 435.35 mL
0.5 mM 8.71 mL 43.54 mL 87.07 mL
1 mM 4.35 mL 21.77 mL 43.54 mL
5 mM 0.87 mL 4.35 mL 8.71 mL

*The above data is based on the productmolecular weight 229.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13236
Actions Antagonist
CAS No. 219911-35-0
Formula C14H11N.HCl
M. Wt 229.7
Purity >98%
Synonyms MPEP hydrochloride
SMILES CC1=CC=CC(=N1)C#CC2=CC=CC=C2.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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