MRGPRX1 agonist 2

Catalog No.: A61588
MRGPRX1 PAM
MRGPRX1 Agonist 2 is a potent positive allosteric modulator of the Mas-related G protein-coupled receptor X1 (MRGPRX1) with an EC50 value of 0.48 μM. This compound is primarily utilized in research focused on neuropathic pain, enabling the exploration of MRGPRX1's role in pain pathways. Its distinct mechanism of action makes it a valuable tool for understanding the modulation of nociceptive signals.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
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Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Biological Activity
DescriptionMRGPRX1 Agonist 2 is a potent positive allosteric modulator of the Mas-related G protein-coupled receptor X1 (MRGPRX1) with an EC50 value of 0.48 μM. This compound is primarily utilized in research focused on neuropathic pain, enabling the exploration of MRGPRX1's role in pain pathways. Its distinct mechanism of action makes it a valuable tool for understanding the modulation of nociceptive signals.
Product Information
Catalog NumA61588
FormulaC15H14N2OS
Molecular Weight270.35
CAS Number302952-43-8
SMILESCC1=CC=CC=C1OC2=C(C(C)=C(C)S3)C3=NC=N2
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