Biological Activity
MRS1706 is a selective adenosine A2B receptor inverse agonist with Ki values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 19.86 mL | 99.29 mL | 198.59 mL |
0.5 mM | 3.97 mL | 19.86 mL | 39.72 mL |
1 mM | 1.99 mL | 9.93 mL | 19.86 mL |
5 mM | 0.4 mL | 1.99 mL | 3.97 mL |
*The above data is based on the productmolecular weight 503.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A16868 |
---|---|
Actions | Agonist |
CAS No. | 264622-53-9 |
Formula | C27H29N5O5 |
M. Wt | 503.56 |
Solubility | DMSO |
Purity | >98% |
Synonyms | MRS 1706, MRS-1706 |
SMILES | O=C(NC1=CC=C(C(C)=O)C=C1)COC2=CC=C(C(N3)=NC(N(CCC)C(N4CCC)=O)=C3C4=O)C=C2 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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