MRS3558

Catalog No.: A57953
A3AR Agonist
MRS3558 is a potent and selective agonist of the A3 adenosine receptor (A3AR), exhibiting Ki values of 0.6 nM for human receptors and 0.9 nM for rat receptors. This compound is valuable for investigating the role of A3AR in neuropathic pain pathways and anesthetic responses. Its high selectivity and potency make it an essential tool for research in receptor pharmacology and therapeutic development.
Grouped product items
Size Price Stock Qty
25mg
$1,780.00
In stock
50mg
$2,280.00
In stock
100mg
$2,960.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionMRS3558 is a potent and selective agonist of the A3 adenosine receptor (A3AR), exhibiting Ki values of 0.6 nM for human receptors and 0.9 nM for rat receptors. This compound is valuable for investigating the role of A3AR in neuropathic pain pathways and anesthetic responses. Its high selectivity and potency make it an essential tool for research in receptor pharmacology and therapeutic development.
Product Information
Catalog NumA57953
FormulaC20H20Cl2N6O3
Molecular Weight463.32
CAS Number793695-40-6
SMILESCNC([C@]12[C@@H]([C@@H](N3C4=NC(Cl)=NC(NCC5=CC(Cl)=CC=C5)=C4N=C3)[C@H](O)[C@@H]2O)C1)=O
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