MRS542

Name: MRS542
Brand: Adooq Bioscience
SKU: A57969
Rating: 5 (288 reviews)

Catalog No.: A57969

A3 AR Antagonist

MRS542 is a nucleoside antagonist of the A3 adenosine receptor (A3 AR) with a pKi of 8.74. In addition to its antagonistic properties, MRS542 functions as a partial agonist, with an effective concentration (pEC50) of 7.76, promoting β-arrestin translocation. This compound is valuable for investigating the role of A3 AR in cardiovascular diseases and related research applications.

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Grouped product items
Size	Price	Stock
25mg	$1,275.00	In stock
50mg	$1,625.00	In stock
100mg	$2,000.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	MRS542 is a nucleoside antagonist of the A3 adenosine receptor (A3 AR) with a pKi of 8.74. In addition to its antagonistic properties, MRS542 functions as a partial agonist, with an effective concentration (pEC50) of 7.76, promoting β-arrestin translocation. This compound is valuable for investigating the role of A3 AR in cardiovascular diseases and related research applications.

Product Information

Catalog Num	A57969
Formula	C17H17ClIN5O4
Molecular Weight	517.71
CAS Number	163152-31-6
SMILES	N(CC1=CC(I)=CC=C1)C2=C3C(N(C=N3)[C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O)=NC(Cl)=N2

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