MS402

Catalog No.: A18866

BRD inhibitor

MS402

MS402 Chemical Structure

CAS NO. 1672684-68-2

MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively.

Availability: In stock

Package Price Qty
5 mg
$350.00
10 mg
$650.00
50 mg
$2,000.00
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Biological Activity

MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.97 mL 134.83 mL 269.67 mL
0.5 mM 5.39 mL 26.97 mL 53.93 mL
1 mM 2.7 mL 13.48 mL 26.97 mL
5 mM 0.54 mL 2.7 mL 5.39 mL

*The above data is based on the productmolecular weight 370.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18866
Actions Inhibitor
CAS No. 1672684-68-2
Formula C20H19ClN2O3
M. Wt 370.83
Purity >98%
Synonyms MS-402, MS 402
SMILES O=C(NC1=CC=C(OC)C=C1)C2=CC=C(NC3=C(C)C(CC3)=O)C(Cl)=C2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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