MS417

Catalog No.: A19433

BRD4 inhibitor

MS417

MS417 Chemical Structure

CAS NO. 916489-36-6

MS417 is a BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM).

Availability: In stock

Package Price Qty
5 mg
$225.00
10 mg
$380.00
50 mg
$940.00
100 mg
$1,600.00
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Biological Activity

MS417 is a BET-specific BRD4 inhibitor, binds to BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively, with weak selectivity at CBP BRD (IC50, 32.7 μM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.1 mL 120.51 mL 241.02 mL
0.5 mM 4.82 mL 24.1 mL 48.2 mL
1 mM 2.41 mL 12.05 mL 24.1 mL
5 mM 0.48 mL 2.41 mL 4.82 mL

*The above data is based on the productmolecular weight 414.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19433
Actions Inhibitor
M. Wt 414.91
Formula C20H19ClN4O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 916489-36-6
Synonyms GTPL-7512, GTPL 7512, GTPL7512, MS 417, MS-417
SMILES O=C(OC)C[[email protected]]1C2=NN=C(C)N2C3=C(C(C)=C(C)S3)C(C4=CC=C(Cl)C=C4)=N1

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