Mu opioid receptor antagonist 3 is a highly potent and selective antagonist of the μ opioid receptor (MOR), with a Ki value of 0.24 nM and an EC50 of 0.54 nM. This compound exhibits strong central nervous system antagonism against morphine and produces fewer withdrawal symptoms compared to traditional antagonists like Naloxone. Mu opioid receptor antagonist 3 is valuable for research applications focused on opioid use disorders (OUD) and studying the mechanisms of opioid dependence and withdrawal.
Mu opioid receptor antagonist 3 is a highly potent and selective antagonist of the μ opioid receptor (MOR), with a Ki value of 0.24 nM and an EC50 of 0.54 nM. This compound exhibits strong central nervous system antagonism against morphine and produces fewer withdrawal symptoms compared to traditional antagonists like Naloxone. Mu opioid receptor antagonist 3 is valuable for research applications focused on opioid use disorders (OUD) and studying the mechanisms of opioid dependence and withdrawal.
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