Nepicastat HCl

Catalog No.: A11172

DBH inhibitor

Nepicastat HCl Chemical Structure

CAS NO. 170151-24-3

Nepicastat hydrochloride is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
50 mg
$300.00
100 mg
$500.00
10mM * 1mL in DMSO
$99.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Nepicastat hydrochloride is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.

Targets
Bovine dopamine-beta-hydroxylase Human dopamine-beta-hydroxylase
8.5 nM9 nM
In vitro DMSO 66 mg/mL (198.9 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.14 mL 150.69 mL 301.38 mL
0.5 mM 6.03 mL 30.14 mL 60.28 mL
1 mM 3.01 mL 15.07 mL 30.14 mL
5 mM 0.6 mL 3.01 mL 6.03 mL

*The above data is based on the productmolecular weight 331.81. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11172
Actions Inhibitor
M. Wt 331.81
Formula C14H15F2N3S.HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 170151-24-3
Synonyms RS-25560-197, SYN117
SMILES C1CC2=C(C=C(C=C2C[[email protected]]1N3C(=CNC3=S)CN)F)F.Cl

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