Olcegepant hydrochloride

Catalog No.: A21900

CGRP1 receptor antagonist

Olcegepant hydrochloride

Olcegepant hydrochloride Chemical Structure

CAS NO. 586368-06-1

Olcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $173.00

Special Price $138.40

10 mg

Regular Price: $298.00

Special Price $238.40

50 mg

Regular Price: $883.00

Special Price $706.40

100 mg

Regular Price: $1,766.00

Special Price $1,412.80

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Biological Activity

Olcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 11.04 mL 55.18 mL 110.36 mL
0.5 mM 2.21 mL 11.04 mL 22.07 mL
1 mM 1.1 mL 5.52 mL 11.04 mL
5 mM 0.22 mL 1.1 mL 2.21 mL

*The above data is based on the productmolecular weight 906.11. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21900
Actions Antagonist
CAS No. 586368-06-1
Formula C38H47Br2N9O5.HCl
M. Wt 906.11
Purity >98%
Synonyms BIBN-4096 hydrochloride, BIBN4096, BIBN 4096; BIBN4096BS hydrochloride, BIBN 4096BS, BIBN-4096BS
SMILES O=C1N(CC2=C(N1)C=CC=C2)C3CCN(C(N[[email protected]@H](C(N[[email protected]](C(N4CCN(C5=CC=NC=C5)CC4)=O)CCCCN)=O)CC6=CC(Br)=C(C(Br)=C6)O)=O)CC3.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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