OP-1074 is a selective estrogen receptor degrader (PA-SERD) that exhibits potent anti-estrogenic activity against both estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ). It effectively inhibits 17β-estradiol (E2)-stimulated transcription, demonstrating IC50 values of 1.6 nM for ERα and 3.2 nM for ERβ. This compound is valuable for research applications focused on hormonal signaling pathways and targeting estrogen-related cancers.
OP-1074 is a selective estrogen receptor degrader (PA-SERD) that exhibits potent anti-estrogenic activity against both estrogen receptor alpha (ERα) and estrogen receptor beta (ERβ). It effectively inhibits 17β-estradiol (E2)-stimulated transcription, demonstrating IC50 values of 1.6 nM for ERα and 3.2 nM for ERβ. This compound is valuable for research applications focused on hormonal signaling pathways and targeting estrogen-related cancers.
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