ORY-1001 (RG-6016)

Catalog No.: A15893

LSD1 Inhibitor

ORY-1001 (RG-6016)

ORY-1001 (RG-6016) Chemical Structure

CAS NO. 1431326-61-2

ORY-1001 is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor with IC50 of <20 nM, with high selectivity against related FAD dependent aminoxidases. Phase 1.

Availability: In stock

Package Price Qty
5 mg
$126.00
10 mg
$214.00
25 mg
$378.00
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Biological Activity

ORY-1001 is an orally active and selective lysine-specific demethylase LSD1/KDM1A inhibitor with IC50 of <20 nM, with high selectivity against related FAD dependent aminoxidases. Phase 1.
Targets
LSD1/KDM1A
20 nM
In vitro DMSO 4 mg/mL (13.18 mM)
Water 53 mg/mL (174.76 mM)
Ethanol Warmed: 3 mg/mL (9.89 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 32.97 mL 164.87 mL 329.74 mL
0.5 mM 6.59 mL 32.97 mL 65.95 mL
1 mM 3.3 mL 16.49 mL 32.97 mL
5 mM 0.66 mL 3.3 mL 6.59 mL

*The above data is based on the productmolecular weight 303.27. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15893
Actions Inhibitor
CAS No. 1431326-61-2
Formula C15H22N2.2HCl
M. Wt 303.27
Purity >98%
Synonyms RG6016, RG-6016
SMILES NC1CCC(N[[email protected]@H]2C[[email protected]]2C3=CC=CC=C3)CC1.Cl.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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