OTX015

Catalog No.: A13890

BET inhibitor

OTX015

OTX015 Chemical Structure

CAS NO. 202590-98-5

OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $70.00

Special Price $63.00

10 mg

Regular Price: $90.00

Special Price $81.00

25 mg

Regular Price: $180.00

Special Price $162.00

50 mg

Regular Price: $250.00

Special Price $225.00

10mM * 1mL in DMSO

Regular Price: $130.00

Special Price $117.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Targets
BRDs (Cell-free assay)
10-19 nM(EC50)
In vitro DMSO 98 mg/mL (199.19 mM)
Water <1 mg/mL (<1 mM)
Ethanol 98 mg/mL (199.19 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.33 mL 101.63 mL 203.26 mL
0.5 mM 4.07 mL 20.33 mL 40.65 mL
1 mM 2.03 mL 10.16 mL 20.33 mL
5 mM 0.41 mL 2.03 mL 4.07 mL

*The above data is based on the productmolecular weight 491.99. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13890
Actions Inhibitor
M. Wt 491.99
Formula C25H22ClN5O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 202590-98-5
Synonyms OTX 015, OTX-015
SMILES CC1=C(SC2=C1C(=N[[email protected]](C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C

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