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Biological Activity
OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Targets
| BRDs (Cell-free assay) | ||||
| 10-19 nM(EC50) |
| In vitro (25°C) | DMSO | 89 mg/mL (180.9 mM) | |
| Water | Insoluble | ||
| Ethanol | 89 mg/mL | ||
| In vivo | 2% DMSO+30% PEG 300+5% Tween 80+ddH2O | 4 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 20.33 mL | 101.63 mL | 203.26 mL |
| 0.5 mM | 4.07 mL | 20.33 mL | 40.65 mL |
| 1 mM | 2.03 mL | 10.16 mL | 20.33 mL |
| 5 mM | 0.41 mL | 2.03 mL | 4.07 mL |
*The above data is based on the productmolecular weight 491.99. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13890 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 202590-98-5 |
| Formula | C25H22ClN5O2S |
| M. Wt | 491.99 |
| Purity | >98% |
| Synonyms | OTX 015, OTX-015 |
| SMILES | CC1=C(SC2=C1C(=N[[email protected]](C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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