OTX015

Catalog No.: A13890
BET inhibitor
OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Grouped product items
Product Name Price Stock Qty
OTX015 5mg
$70.00
In stock
OTX015 10mg
$90.00
In stock
OTX015 25mg
$180.00
In stock
OTX015 50mg
$250.00
In stock
OTX015 10mM * 1mL in DMSO
$130.00
In stock
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Adooq Products cited in reputable paper
Biological Activity
Discription OTX015 is an orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM).
Targets
Target Value
Product Information
Catalog Num A13890
Formula C25H22ClN5O2S
Molecular Weight 491.99
CAS Number 202590-98-5
SMILES CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C
Synonyms OTX 015, OTX-015
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro (25°C) DMSO 89 mg/mL (180.9 mM)
Water Insoluble
Ethanol 89 mg/mL
In vivo 2% DMSO+30% PEG 300+5% Tween 80+ddH2O 4 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.33 mL 101.63 mL 203.26 mL
0.5 mM 4.07 mL 20.33 mL 40.65 mL
1 mM 2.03 mL 10.16 mL 20.33 mL
5 mM 0.41 mL 2.03 mL 4.07 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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