PROTAC ERα Degrader-5 (PAC)

Name: PROTAC ERα Degrader-5 (PAC)
Brand: Adooq Bioscience
SKU: A12939
Rating: 5 (288 reviews)

Catalog No.: A12939

PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab).

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PROTAC ERα Degrader-5 (PAC) 2158322-33-7

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Grouped product items
Size	Price	Stock
1mg	$820.00	In stock
5mg	$1,820.00	In stock
10mg	$2,980.00	In stock
50mg	$9,820.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	PAC, consists the ADCs linker and PROTACs, conjugated to an antibody. PAC extracts from patent WO2017201449A1, compound LP2. PAC conjugated to an antibody is a more marked estrogen receptor-alpha (ERα) degrader compared to PROTAC (without Ab).

Product Information

Catalog Num	A12939
Formula	C94H107N13O16
Molecular Weight	1674.93
CAS Number	2158322-33-7
SMILES	CN(C(COCCOCCNC(C1=CC=C(C(N2[C@@H](C)[C@H](NC([C@H](C)NC)=O)C(N(CC3=C(OC)C=CC4=C3C=CC=C4)C5=C2C=C(C#N)C=C5)=O)=O)C=C1)=O)=O)CCOC(C=C6)=CC=C6/C(C7=CC=C(OCC(C=C8)=CC=C8NC([C@H](CCCNC(N)=O)NC([C@H](C(C)C)NC(CCCCCN9C(C=CC9=O)=O)=O)=O)=O)C=C7)=C(C%10=CC=CC=C%10)/CC
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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