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PF 4981517

CYP3A4 inhibitor

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Catalog No. A12544

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
PF 4981517 5mg A12544-5
PF 4981517 10mg A12544-10
PF 4981517 25mg A12544-25
PF 4981517 50mg A12544-50
PF 4981517 10mM * 1mL in DMSO A12544-10mM-D

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).

PF 4981517

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Chemical Information

Catalog Num A12544
Actions Inhibitor
M. Wt 456.59
Formula C26H32N8
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1390637-82-7
Synonyms PF4981517, PF-4981517
SMILES CC1=CC=C(C=C1)C2=C(C=NN2C)C3=NN(C4=C3C(=NC=N4)N5CC[[email protected]@H](C5)N6CCCCC6)C

Biological Activity

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).
30 nM


Solubility (25°C)* In vitro DMSO 91 mg/mL (199.3 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.9 mL 109.51 mL 219.01mL
0.5 mM 4.38 mL 21.9 mL 43.8 mL
1 mM 2.19 mL 10.95 mL 21.9 mL
5 mM 0.44 mL 2.19 mL 4.38 mL

*The above data is based on the productmolecular weight 456.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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