PF 4981517

Name: PF 4981517
SKU: A12544
Price: 64 USD
Rating: 5 (288 reviews)

Catalog No.: A12544

CYP3A4 inhibitor

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).

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Grouped product items
Product Name	Price	Stock
PF 4981517 5mg	Special Price $64.00 Regular Price $80.00	In stock
PF 4981517 10mg	Special Price $112.00 Regular Price $140.00	In stock
PF 4981517 25mg	Special Price $224.00 Regular Price $280.00	In stock
PF 4981517 50mg	Special Price $400.00 Regular Price $500.00	In stock
*PF 4981517 10mM 1mL in DMSO**	Special Price $105.60 Regular Price $132.00	In stock
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Data Sheet

SDS

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Biological Activity

Discription

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).

Targets

Target	Value

Product Information

Catalog Num	A12544
Formula	C26H32N8
Molecular Weight	456.59
CAS Number	1390637-82-7
SMILES	CC1=CC=C(C=C1)C2=C(C=NN2C)C3=NN(C4=C3C(=NC=N4)N5CC[C@@H](C5)N6CCCCC6)C
Synonyms	PF4981517, PF-4981517
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	85 mg/mL (186.16 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.9 mL	109.51 mL	219.01 mL
0.5 mM	4.38 mL	21.9 mL	43.8 mL
1 mM	2.19 mL	10.95 mL	21.9 mL
5 mM	0.44 mL	2.19 mL	4.38 mL

Useful Calculator

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