PF 4981517

Catalog No.: A12544

CYP3A4 inhibitor

PF 4981517

PF 4981517 Chemical Structure

CAS NO. 1390637-82-7

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).

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5 mg

Regular Price: $80.00

Special Price $64.00

10 mg

Regular Price: $140.00

Special Price $112.00

25 mg

Regular Price: $280.00

Special Price $224.00

50 mg

Regular Price: $500.00

Special Price $400.00

10mM * 1mL in DMSO

Regular Price: $132.00

Special Price $105.60

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Biological Activity

PF 4981517 is a potent and selective inhibitor of CYP3A4 (IC50 values are 0.03, 17 and 70 μM for CYP3A4, CYP3A5 and CYP3A7 respectively).
Targets
CYP3A4
30 nM
In vitro DMSO 85 mg/mL (186.16 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.9 mL 109.51 mL 219.01 mL
0.5 mM 4.38 mL 21.9 mL 43.8 mL
1 mM 2.19 mL 10.95 mL 21.9 mL
5 mM 0.44 mL 2.19 mL 4.38 mL

*The above data is based on the productmolecular weight 456.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12544
Actions Inhibitor
CAS No. 1390637-82-7
Formula C26H32N8
M. Wt 456.59
Purity >98%
Synonyms PF4981517, PF-4981517
SMILES CC1=CC=C(C=C1)C2=C(C=NN2C)C3=NN(C4=C3C(=NC=N4)N5CC[[email protected]@H](C5)N6CCCCC6)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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