PF-CBP1

Catalog No.: A15876

CREBBP inhibitor

PF-CBP1

PF-CBP1 Chemical Structure

CAS NO. 1962928-21-7

PF-CBP1 is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.

Availability: In stock

Package Price Qty
10 mg
$80.00
25 mg
$180.00
50 mg
$300.00
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Biological Activity

PF-CBP1 is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.47 mL 102.33 mL 204.67 mL
0.5 mM 4.09 mL 20.47 mL 40.93 mL
1 mM 2.05 mL 10.23 mL 20.47 mL
5 mM 0.41 mL 2.05 mL 4.09 mL

*The above data is based on the productmolecular weight 488.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15876
Actions Inhibitor
CAS No. 1962928-21-7
Formula C29H36N4O3
M. Wt 488.6
Purity >98%
Synonyms PF-CBP-1, PF-CBP 1, PF-06670910, PF 06670910, PF06670910
SMILES CCCOC1=CC=C(C=C1)CCC2=NC3=C(N2CCN4CCOCC4)C=CC(=C3)C5=C(ON=C5C)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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