PFK-158

Catalog No.: A14398

PFK-2/FBPase inhibitor

PFK-158

PFK-158 Chemical Structure

CAS NO. 1462249-75-7

PFK-158 is an inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatases (PFK-2/FBPase) isoform 3 (PFKFB3) and derivative of 3-(3-pyridinyl)-1-[4-pyridinyl]-2-propen-1-one (3PO), with potential antineoplastic activity.

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Package Price Qty
5 mg
$55.00
10 mg
$90.00
25 mg
$190.00
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Biological Activity

PFK-158 is an inhibitor of 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatases (PFK-2/FBPase) isoform 3 (PFKFB3) and derivative of 3-(3-pyridinyl)-1-[4-pyridinyl]-2-propen-1-one (3PO), with potential antineoplastic activity.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.46 mL 152.3 mL 304.61 mL
0.5 mM 6.09 mL 30.46 mL 60.92 mL
1 mM 3.05 mL 15.23 mL 30.46 mL
5 mM 0.61 mL 3.05 mL 6.09 mL

*The above data is based on the productmolecular weight 328.29. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14398
Actions Inhibitor
M. Wt 328.29
Formula C18H11F3N2O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1462249-75-7
Synonyms PFK 158, PFK158, ACT-PEK-158
SMILES O=C(C1=CC=NC=C1)/C=C/C2=NC3=CC(C(F)(F)F)=CC=C3C=C2

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