Pitolisant hydrochloride

Catalog No.: A15213

Nonimidazole inverse agonist

Pitolisant hydrochloride

Pitolisant hydrochloride Chemical Structure

CAS NO. 903576-44-3

Pitolisant hydrochloride is a novel, potent, and selective nonimidazole inverse agonist at the recombinant human H3 receptor (Ki=0.16 nM).

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10 mg

Regular Price: $90.00

Special Price $72.00

50 mg

Regular Price: $400.00

Special Price $320.00

100 mg

Regular Price: $680.00

Special Price $544.00

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Biological Activity

Pitolisant hydrochloride is a novel, potent, and selective nonimidazole inverse agonist at the recombinant human H3 receptor (Ki=0.16 nM).
In vitro DMSO 57 mg/mL (171.52 mM)
Water 57 mg/mL (171.52 mM)
Ethanol 57 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.09 mL 150.46 mL 300.92 mL
0.5 mM 6.02 mL 30.09 mL 60.18 mL
1 mM 3.01 mL 15.05 mL 30.09 mL
5 mM 0.6 mL 3.01 mL 6.02 mL

*The above data is based on the productmolecular weight 332.31. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15213
Actions Agonist
CAS No. 903576-44-3
Formula C17H27Cl2NO
M. Wt 332.31
Purity >98%
Synonyms Ciproxidine, BF 2649, BF2649, BF-2649
SMILES C1CCN(CC1)CCCOCCCC2=CC=C(C=C2)Cl.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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