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PKR Inhibitor is an oxindole/imidazole derivative that binds the ATP-binding site of PKR and blocks autophosphorylation with an IC50 value of 186-210 nM.3 PKR Inhibitor protects human neuroblastoma cells against cell damage triggered by tunicamycin-mediated endoplasmic reticulum stress.
| In vitro | DMSO | 13 mg/mL (48.45 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 37.27 mL | 186.36 mL | 372.72 mL |
| 0.5 mM | 7.45 mL | 37.27 mL | 74.54 mL |
| 1 mM | 3.73 mL | 18.64 mL | 37.27 mL |
| 5 mM | 0.75 mL | 3.73 mL | 7.45 mL |
*The above data is based on the productmolecular weight 268.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13538 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 608512-97-6 |
| Formula | C13H8N4OS |
| M. Wt | 268.3 |
| Purity | >98% |
| Synonyms | C16, GW 506033X |
| SMILES | C1=CC2=C(C\3=C1NC(=O)/C3=C\C4=CN=CN4)SC=N2 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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