PROTAC BET degrader-2

Catalog No.: A18785

PROTAC BET degrader

PROTAC BET degrader-2

PROTAC BET degrader-2 Chemical Structure

CAS NO. 2093388-33-9

PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression.

Availability: In stock

Package Price Qty
5 mg
$450.00
10 mg
$775.00
50 mg
$2,300.00
100 mg
$4,600.00
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Biological Activity

PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.97 mL 64.86 mL 129.73 mL
0.5 mM 2.59 mL 12.97 mL 25.95 mL
1 mM 1.3 mL 6.49 mL 12.97 mL
5 mM 0.26 mL 1.3 mL 2.59 mL

*The above data is based on the productmolecular weight 770.84. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18785
Actions Degrader
CAS No. 2093388-33-9
Formula C41H42N10O6
M. Wt 770.84
Solubility DMSO
Purity >98%
SMILES O=C(C1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1)NCCCC7=CC=CC8=C7CN(C(CC9)C(NC9=O)=O)C8=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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