PROTAC BRD4 ligand-2

Catalog No.: A40601
Ligands for Target Protein for PROTAC Chemical
PROTAC BRD4 ligand-2 is a specific ligand for the BRD4 protein, designed for use in PROTAC-mediated degradation strategies. This compound facilitates the targeted degradation of BRD4, a key regulator of transcription and associated with various cancers, by recruiting the E3 ubiquitin ligase. It is instrumental in research applications aimed at understanding BRD4's role in oncogenesis and therapeutic development in cancer treatments.
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Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Biological Activity
DescriptionPROTAC BRD4 ligand-2 is a specific ligand for the BRD4 protein, designed for use in PROTAC-mediated degradation strategies. This compound facilitates the targeted degradation of BRD4, a key regulator of transcription and associated with various cancers, by recruiting the E3 ubiquitin ligase. It is instrumental in research applications aimed at understanding BRD4's role in oncogenesis and therapeutic development in cancer treatments.
Product Information
Catalog NumA40601
FormulaC22H17ClN6
Molecular Weight400.86
CAS Number2154358-11-7
SMILESClC1=CC=C(C2=NC3(CC3)C4=NN=C(C)N4C5=CC=C(C6=CNN=C6)C=C25)C=C1
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