Proxyfan is a potent antagonist of the histamine H3 receptor, exhibiting Ki values of 2.9 nM and 2.7 nM for rat and human H3 receptors, respectively. This compound demonstrates over 1000-fold selectivity for the H3 receptor compared to other histamine receptors. Proxyfan is useful in research applications focused on neurological disorders, cognitive enhancement, and sleep regulation, making it a valuable tool for studying histaminergic signaling pathways.
Proxyfan is a potent antagonist of the histamine H3 receptor, exhibiting Ki values of 2.9 nM and 2.7 nM for rat and human H3 receptors, respectively. This compound demonstrates over 1000-fold selectivity for the H3 receptor compared to other histamine receptors. Proxyfan is useful in research applications focused on neurological disorders, cognitive enhancement, and sleep regulation, making it a valuable tool for studying histaminergic signaling pathways.
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