Proxyphylline

Catalog No.: A16821
A1 adenosine receptors antagonist
Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets).
Grouped product items
Product Name Price Stock Qty
Proxyphylline 100mg
$50.00
In stock
Proxyphylline 200mg
$80.00
In stock
Proxyphylline 500mg
$150.00
In stock
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Biological Activity
Discription Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets).
Product Information
Catalog Num A16821
Formula C10H14N4O3
Molecular Weight 238.25
CAS Number 603-00-9
SMILES CC(CN1C=NC2=C1C(=O)N(C(=O)N2C)C)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility
In vitro DMSO 42 mg/mL (176.29 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 41.97 mL 209.86 mL 419.73 mL
0.5 mM 8.39 mL 41.97 mL 83.95 mL
1 mM 4.2 mL 20.99 mL 41.97 mL
5 mM 0.84 mL 4.2 mL 8.39 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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