Proxyphylline

Name: Proxyphylline
Brand: Adooq Bioscience
SKU: A16821
Rating: 5 (288 reviews)

Catalog No.: A16821

A1 adenosine receptors antagonist

Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets).

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Proxyphylline 603-00-9 A1 adenosine receptors antagonist

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Grouped product items
Size	Price	Stock
200mg	$20.00	In stock
500mg	$35.00	In stock
*10mM 1mL in DMSO**	$40.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Adooq Products cited in reputable paper

Biological Activity

Description	Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets).

Product Information

Catalog Num	A16821
Formula	C10H14N4O3
Molecular Weight	238.25
CAS Number	603-00-9
SMILES	CC(CN1C=NC2=C1C(=O)N(C(=O)N2C)C)O
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	42 mg/mL (176.29 mM)
	* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	41.97 mL	209.86 mL	419.73 mL
0.5 mM	8.39 mL	41.97 mL	83.95 mL
1 mM	4.2 mL	20.99 mL	41.97 mL
5 mM	0.84 mL	4.2 mL	8.39 mL

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