Biological Activity
(R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM).
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 28.49 mL | 142.45 mL | 284.89 mL |
0.5 mM | 5.7 mL | 28.49 mL | 56.98 mL |
1 mM | 2.85 mL | 14.24 mL | 28.49 mL |
5 mM | 0.57 mL | 2.85 mL | 5.7 mL |
*The above data is based on the productmolecular weight 351.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21358 |
---|---|
Actions | Inhibitor |
CAS No. | 1593478-56-8 |
Formula | C11H10Br2FNO |
M. Wt | 351.01 |
Solubility | DMSO |
Purity | >98% |
SMILES | O=CN1[[email protected]](C)CCC2=C1C=C(Br)C(F)=C2Br |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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