Relugolix

Catalog No.: A17783

GnRH antagonist

Relugolix

Relugolix Chemical Structure

CAS NO. 737789-87-6

Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013.

Availability: In stock

Package Price Qty
1 mg
$60.00
5 mg
$110.00
10 mg
$180.00
50 mg
$600.00
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Biological Activity

Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.04 mL 80.18 mL 160.35 mL
0.5 mM 3.21 mL 16.04 mL 32.07 mL
1 mM 1.6 mL 8.02 mL 16.04 mL
5 mM 0.32 mL 1.6 mL 3.21 mL

*The above data is based on the productmolecular weight 623.63. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A17783
Actions Antagonist
M. Wt 623.63
Formula C29H27F2N7O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 737789-87-6
Synonyms TAK385; TAK-385; TAK 385; Relugolix.
SMILES O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1

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