RPR-260243

Catalog No.: A20977

HERG activator

RPR-260243

RPR-260243 Chemical Structure

CAS NO. 668463-35-2

RPR-260243 is a novel activator of HERG; modifies HERG currents inhibited by dofetilide (IC50 = 58 nM); little effect on HERG current amplitude and no significant effects on steady-state activation parameters or on channel inactivation processes.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $238.00

Special Price $190.40

10 mg

Regular Price: $409.00

Special Price $327.20

50 mg

Regular Price: $1,214.00

Special Price $971.20

100 mg

Regular Price: $2,429.00

Special Price $1,943.20

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Biological Activity

RPR-260243 is a novel activator of HERG; modifies HERG currents inhibited by dofetilide (IC50 = 58 nM); little effect on HERG current amplitude and no significant effects on steady-state activation parameters or on channel inactivation processes.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.59 mL 97.94 mL 195.89 mL
0.5 mM 3.92 mL 19.59 mL 39.18 mL
1 mM 1.96 mL 9.79 mL 19.59 mL
5 mM 0.39 mL 1.96 mL 3.92 mL

*The above data is based on the productmolecular weight 510.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A20977
Actions Activator
CAS No. 668463-35-2
Formula C28H25F3N2O4
M. Wt 510.5
Purity >98%
Synonyms RPR260243, RPR 260243
SMILES O=C([[email protected]]1CN(CC#CC2=CC(F)=CC(F)=C2F)CC[[email protected]]1CCC(C3=CC=NC4=CC=C(OC)C=C34)=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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