RS 17053 HCl

Catalog No.: A16885

α1A antagonist

RS 17053 HCl

RS 17053 HCl Chemical Structure

CAS NO. 169505-93-5

RS 17053 HCl is α1A-adrenoceptor antagonist, with very high affinity for α1A receptors (pKi and pA2 estimates of 9.1 - 9.9) and a 30 - 100 fold selectivity over the α1B and α1D subtypes (pKi and pA2 estimates 7.7 - 7.8).

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
50 mg
$380.00
100 mg
$700.00
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Biological Activity

RS 17053 HCl is α1A-adrenoceptor antagonist, with very high affinity for α1A receptors (pKi and pA2 estimates of 9.1 - 9.9) and a 30 - 100 fold selectivity over the α1B and α1D subtypes (pKi and pA2 estimates 7.7 - 7.8).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.25 mL 111.25 mL 222.51 mL
0.5 mM 4.45 mL 22.25 mL 44.5 mL
1 mM 2.23 mL 11.13 mL 22.25 mL
5 mM 0.45 mL 2.23 mL 4.45 mL

*The above data is based on the productmolecular weight 449.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16885
Actions Antagonist
M. Wt 449.42
Formula C24H29N2O2Cl?HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 169505-93-5
Synonyms RS-17053, RS17053
SMILES Cl.CC(C)(CC1=CNC2=CC=C(Cl)C=C12)NCCOC1=C(OCC2CC2)C=CC=C1

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