Rupatadine Fumarate

Catalog No.: A12356

PAFR inhibitor/H1 receptor inhibitor

Rupatadine Fumarate

Rupatadine Fumarate Chemical Structure

CAS NO. 182349-12-8

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $60.00

Special Price $54.00

10 mg

Regular Price: $100.00

Special Price $90.00

25 mg

Regular Price: $200.00

Special Price $180.00

50 mg

Regular Price: $350.00

Special Price $315.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.
Targets
Histamine H1 receptor PAFR
102 nM(Ki)550 nM(Ki)
In vitro (25°C) DMSO 9 mg/mL (16.91 mM)
Water <1 mg/mL (<1 mM)
Ethanol 13 mg/mL (24.43 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.8 mL 93.98 mL 187.96 mL
0.5 mM 3.76 mL 18.8 mL 37.59 mL
1 mM 1.88 mL 9.4 mL 18.8 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 532.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A12356
Actions Inhibitor
M. Wt 532.03
Formula C26H26ClN3.C4H4O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 182349-12-8
Synonyms N/A
SMILES CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O

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