Rupatadine Fumarate

Catalog No.: A12356

PAFR inhibitor/H1 receptor inhibitor

Rupatadine Fumarate

Rupatadine Fumarate Chemical Structure

CAS NO. 182349-12-8

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.

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100 mg
$86.00
500 mg
$200.00
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Biological Activity

Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 and 102 nM, respectively.
Targets
Histamine H1 receptor PAFR
102 nM(Ki)550 nM(Ki)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.8 mL 93.98 mL 187.96 mL
0.5 mM 3.76 mL 18.8 mL 37.59 mL
1 mM 1.88 mL 9.4 mL 18.8 mL
5 mM 0.38 mL 1.88 mL 3.76 mL

*The above data is based on the productmolecular weight 532.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12356
Actions Inhibitor
CAS No. 182349-12-8
Formula C26H26ClN3.C4H4O4
M. Wt 532.03
Purity >98%
SMILES CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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