S1RA

Catalog No.: A12504

sigma-1 receptor antagonist

S1RA Chemical Structure

CAS NO. 878141-96-9

S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ± 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.

Availability: In stock

Package Price Qty
5 mg
$350.00
10 mg
$540.00
25 mg
$1,000.00
50 mg
$1,620.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ± 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.64 mL 148.18 mL 296.37 mL
0.5 mM 5.93 mL 29.64 mL 59.27 mL
1 mM 2.96 mL 14.82 mL 29.64 mL
5 mM 0.59 mL 2.96 mL 5.93 mL

*The above data is based on the productmolecular weight 337.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12504
Actions Antagonist
M. Wt 337.42
Formula C20H23N3O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 878141-96-9
Synonyms E-52862
SMILES CC1=CC(=NN1C2=CC3=CC=CC=C3C=C2)OCCN4CCOCC4

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