SA-4503

Catalog No.: A12984

sigma 1 receptor(σ1R) agonist

SA-4503

SA-4503 Chemical Structure

CAS NO. 165377-44-6

SA4503 is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50 = 17.4 +/- 1.9 nM); 100-fold less affinity for the sigma 2 receptor.

Availability: In stock

Package Price Qty
10 mg
$120.00
50 mg
$500.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

SA4503 is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50 = 17.4 +/- 1.9 nM); 100-fold less affinity for the sigma 2 receptor.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.65 mL 113.27 mL 226.54 mL
0.5 mM 4.53 mL 22.65 mL 45.31 mL
1 mM 2.27 mL 11.33 mL 22.65 mL
5 mM 0.45 mL 2.27 mL 4.53 mL

*The above data is based on the productmolecular weight 441.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A12984
Actions Agonist
M. Wt 441.43
Formula C23H32N2O2.2HCl
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 165377-44-6
Synonyms AGY-94806, AGY94806, AGY 94806Cutamesine
SMILES COC1=C(OC)C=CC(CCN2CCN(CCCC3=CC=CC=C3)CC2)=C1.Cl.Cl

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