SA-4503

Catalog No.: A12984

sigma 1 receptor(σ1R) agonist

SA-4503

SA-4503 Chemical Structure

CAS NO. 165377-44-6

SA4503 is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50 = 17.4 +/- 1.9 nM); 100-fold less affinity for the sigma 2 receptor.

Availability: In stock

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10 mg

Regular Price: $120.00

Special Price $96.00

50 mg

Regular Price: $500.00

Special Price $400.00

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Biological Activity

SA4503 is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50 = 17.4 +/- 1.9 nM); 100-fold less affinity for the sigma 2 receptor.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.65 mL 113.27 mL 226.54 mL
0.5 mM 4.53 mL 22.65 mL 45.31 mL
1 mM 2.27 mL 11.33 mL 22.65 mL
5 mM 0.45 mL 2.27 mL 4.53 mL

*The above data is based on the productmolecular weight 441.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12984
Actions Agonist
CAS No. 165377-44-6
Formula C23H32N2O2.2HCl
M. Wt 441.43
Purity >98%
Synonyms AGY-94806, AGY94806, AGY 94806Cutamesine
SMILES COC1=C(OC)C=CC(CCN2CCN(CCCC3=CC=CC=C3)CC2)=C1.Cl.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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