Biological Activity
SA4503 is a selective sigma 1 receptor(σ1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50 = 17.4 +/- 1.9 nM); 100-fold less affinity for the sigma 2 receptor.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.65 mL | 113.27 mL | 226.54 mL |
0.5 mM | 4.53 mL | 22.65 mL | 45.31 mL |
1 mM | 2.27 mL | 11.33 mL | 22.65 mL |
5 mM | 0.45 mL | 2.27 mL | 4.53 mL |
*The above data is based on the productmolecular weight 441.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A12984 |
---|---|
Actions | Agonist |
CAS No. | 165377-44-6 |
Formula | C23H32N2O2.2HCl |
M. Wt | 441.43 |
Purity | >98% |
Synonyms | AGY-94806, AGY94806, AGY 94806Cutamesine |
SMILES | COC1=C(OC)C=CC(CCN2CCN(CCCC3=CC=CC=C3)CC2)=C1.Cl.Cl |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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