Biological Activity
SB 242084 is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.33 mL | 126.63 mL | 253.26 mL |
0.5 mM | 5.07 mL | 25.33 mL | 50.65 mL |
1 mM | 2.53 mL | 12.66 mL | 25.33 mL |
5 mM | 0.51 mL | 2.53 mL | 5.07 mL |
*The above data is based on the productmolecular weight 394.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21715 |
---|---|
Actions | Antagonist |
CAS No. | 181632-25-7 |
Formula | C21H19ClN4O2 |
M. Wt | 394.85 |
Solubility | DMSO |
Purity | >98% |
Synonyms | SB-242084, SB242084 |
SMILES | O=C(N1CCC2=C1C=C(Cl)C(C)=C2)NC3=CC=C(OC4=CC=CN=C4C)N=C3 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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