Biological Activity
SB408124 Hcl is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively; exhibits 50-fold selectivity over OX2 receptor.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.46 mL | 127.28 mL | 254.56 mL |
0.5 mM | 5.09 mL | 25.46 mL | 50.91 mL |
1 mM | 2.55 mL | 12.73 mL | 25.46 mL |
5 mM | 0.51 mL | 2.55 mL | 5.09 mL |
*The above data is based on the productmolecular weight 392.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A15231 |
---|---|
Actions | Antagonist |
M. Wt | 392.83 |
Formula | C19H19ClF2N4O |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1431697-90-3 |
Synonyms | SB 408124 Hydrochloride, SB408124 Hydrochloride |
SMILES | CC1=NC2=C(C=C(C=C2C(=C1)NC(=O)NC3=CC=C(C=C3)N(C)C)F)F.Cl |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy SB-408124 HCl | SB-408124 HCl Supplier | purchase | cost | manufacturer | order | distributor | buy 1431697-90-3| 1431697-90-3 Supplier | purchase 1431697-90-3 | 1431697-90-3 cost | 1431697-90-3 manufacturer | order 1431697-90-3 | 1431697-90-3 distributor