SB-674042

Catalog No.: A15233

OX1 receptor antagonist

SB-674042

SB-674042 Chemical Structure

CAS NO. 483313-22-0

SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM); exhibits 100-fold selectivity for OX1 over OX2 receptors.

Availability: In stock

Package Price Qty
5 mg
$94.00
10 mg
$160.00
50 mg
$480.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM); exhibits 100-fold selectivity for OX1 over OX2 receptors.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.3 mL 111.48 mL 222.96 mL
0.5 mM 4.46 mL 22.3 mL 44.59 mL
1 mM 2.23 mL 11.15 mL 22.3 mL
5 mM 0.45 mL 2.23 mL 4.46 mL

*The above data is based on the productmolecular weight 448.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15233
Actions Antagonist
M. Wt 448.51
Formula C24H21FN4O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 483313-22-0
Synonyms SB 674042, SB674042
SMILES CC1=NC(=C(S1)C2=CC=CC=C2F)C(=O)N3CCCC3CC4=NN=C(O4)C5=CC=CC=C5

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