SB-674042

Catalog No.: A15233

OX1 receptor antagonist

SB-674042

SB-674042 Chemical Structure

CAS NO. 483313-22-0

SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM); exhibits 100-fold selectivity for OX1 over OX2 receptors.

Availability: In stock

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5 mg

Regular Price: $94.00

Special Price $75.20

10 mg

Regular Price: $160.00

Special Price $128.00

50 mg

Regular Price: $480.00

Special Price $384.00

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Biological Activity

SB-674042 is a potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM); exhibits 100-fold selectivity for OX1 over OX2 receptors.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.3 mL 111.48 mL 222.96 mL
0.5 mM 4.46 mL 22.3 mL 44.59 mL
1 mM 2.23 mL 11.15 mL 22.3 mL
5 mM 0.45 mL 2.23 mL 4.46 mL

*The above data is based on the productmolecular weight 448.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15233
Actions Antagonist
CAS No. 483313-22-0
Formula C24H21FN4O2S
M. Wt 448.51
Purity >98%
Synonyms SB 674042, SB674042
SMILES CC1=NC(=C(S1)C2=CC=CC=C2F)C(=O)N3CCCC3CC4=NN=C(O4)C5=CC=CC=C5
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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