SB-742457

Catalog No.: A14092

5-HT6 receptor antagonist

SB-742457

SB-742457 Chemical Structure

CAS NO. 607742-69-8

SB-742457 is a selective 5-HT6 receptor antagonist with cognition, memory, and learning-enhancing effects.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $90.00

Special Price $81.00

10 mg

Regular Price: $150.00

Special Price $135.00

25 mg

Regular Price: $300.00

Special Price $270.00

10mM * 1mL in DMSO

Regular Price: $120.00

Special Price $108.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

SB-742457 is a selective 5-HT6 receptor antagonist with cognition, memory, and learning-enhancing effects.
Targets
5-HT6
9.63(pKi)
In vitro (25°C) DMSO 78 mg/mL (220.68 mM)
Water <1 mg/mL (<1 mM)
Ethanol 2 mg/mL (5.65 mM)
In vivo 2% DMSO, 48% PEG300, 2% Tween 80 and 48% water 5 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.29 mL 141.47 mL 282.93 mL
0.5 mM 5.66 mL 28.29 mL 56.59 mL
1 mM 2.83 mL 14.15 mL 28.29 mL
5 mM 0.57 mL 2.83 mL 5.66 mL

*The above data is based on the productmolecular weight 353.444. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14092
Actions Antagonist
M. Wt 353.444
Formula C19H19N3O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 607742-69-8
Synonyms GSK 742457, SB742457, SB 742457, GSK742457, SB-742,457
SMILES C1CN(CCN1)C2=CC=CC3=CC(=CN=C32)S(=O)(=O)C4=CC=CC=C4

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