SCH 442416

Name: SCH 442416
SKU: A12695
Price: 96 USD
Rating: 5 (288 reviews)

Catalog No.: A12695

A2A Receptor Antagonist

SCH 442416 is a selective adenosine A2A receptor antagonist; binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).

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Grouped product items
Product Name	Stock
SCH 442416 10mg	Please Inquiry
SCH 442416 25mg	Please Inquiry
SCH 442416 50mg	Please Inquiry
SCH 442416 100mg	Please Inquiry
Bulk Size	Bulk Discount

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Data Sheet

SDS

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Biological Activity

Discription	SCH 442416 is a selective adenosine A2A receptor antagonist; binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).

Product Information

Catalog Num	A12695
Formula	C20H19N7O2
Molecular Weight	389.42
CAS Number	316173-57-6
SMILES	COC1=CC=C(C=C1)CCCN2C3=C(C=N2)C4=NC(=NN4C(=N3)N)C5=CC=CO5
Synonyms	SCH442416, SCH-442416
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	72 mg/mL (184.89 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.68 mL	128.4 mL	256.79 mL
0.5 mM	5.14 mL	25.68 mL	51.36 mL
1 mM	2.57 mL	12.84 mL	25.68 mL
5 mM	0.51 mL	2.57 mL	5.14 mL

Useful Calculator

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