SCH 442416

Catalog No.: A12695

A2A Receptor Antagonist

SCH 442416

SCH 442416 Chemical Structure

CAS NO. 316173-57-6

SCH 442416 is a selective adenosine A2A receptor antagonist; binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).

Availability: In stock

Package Price Qty
10 mg
$120.00
25 mg
$240.00
50 mg
$480.00
100 mg
$900.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

SCH 442416 is a selective adenosine A2A receptor antagonist; binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). Displays > 23000-fold selectivity for hA2A over hA1 in vitro with minimal affinity for hA2B and hA3 receptors (IC50 > 10 μM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.68 mL 128.4 mL 256.79 mL
0.5 mM 5.14 mL 25.68 mL 51.36 mL
1 mM 2.57 mL 12.84 mL 25.68 mL
5 mM 0.51 mL 2.57 mL 5.14 mL

*The above data is based on the productmolecular weight 389.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12695
Actions Antagonist
M. Wt 389.42
Formula C20H19N7O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 316173-57-6
Synonyms SCH442416, SCH-442416
SMILES COC1=CC=C(C=C1)CCCN2C3=C(C=N2)C4=NC(=NN4C(=N3)N)C5=CC=CO5

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