SCH772984

Name: SCH772984
SKU: A12824
Price: 40 USD
Rating: 5 (6 reviews)

Catalog No.: A12824

ERK Inhibitor

Adooq's SCH772984 has been cited by 6 publications

SCH772984 is a novel, specific inhibitor of ERK1/2 with IC50 of 4 nM and 1 nM, respectively.

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Grouped product items
Size	Price	Stock
1mg	$40.00	In stock
2mg	$65.00	In stock
5mg	$85.00	In stock
10mg	$135.00	In stock
25mg	$295.00	In stock
50mg	$445.00	In stock
100mg	$670.00	In stock
200mg	$955.00	In stock
500mg	$1,425.00	In stock
*10mM 1mL in DMSO**	$125.00	In stock
Bulk Size	Bulk Discount

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

Adooq Products cited in reputable paper

Adooq's SCH772984 has been cited by 6 publications

Yuki Shimizu, .et al. , Cancer Lett, 2022, Sep 1;543 PMID: 35724767

Yajun Li, .et al. , Cell Prolif, 2022, Oct;55(10) PMID: 35708050

Sergey A. Dyshlovoy, .et al. , Pharmaceuticals, 2021, 14(10), 949

Sergey A Dyshlovoy, .et al. , Sci Rep, 2020, Aug 6;10(1):13178 PMID: 32764580

Guo X, .et al. , Pflugers Arch, 2018, Jun;470(6):909-921 PMID: 29441404

Takuya Hasegawa, .et al. , FEBS Open Bio, 2017, Aug; 7(8): 1154-1165 PMID: 28781955

Biological Activity

Discription

SCH772984 is a novel, specific inhibitor of ERK1/2 with IC50 of 4 nM and 1 nM, respectively.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

Product Information

Catalog Num	A12824
Formula	C33H33N9O2
Molecular Weight	587.68
CAS Number	942183-80-4
SMILES	C1CN(C[C@@H]1C(=O)NC2=CC3=C(C=C2)NN=C3C4=CC=NC=C4)CC(=O)N5CCN(CC5)C6=CC=C(C=C6)C7=NC=CC=N7
Synonyms	SCH-772984, SCH 772984
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro (25°C)	DMSO	Warmed: 13 mg/mL (22.12 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	5% DMSO+30% PEG 300+ddH2O	0.5 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.02 mL	85.08 mL	170.16 mL
0.5 mM	3.4 mL	17.02 mL	34.03 mL
1 mM	1.7 mL	8.51 mL	17.02 mL
5 mM	0.34 mL	1.7 mL	3.4 mL

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