SGC 707

Catalog No.: A15450

PRMT3 Inhibitor

SGC 707

SGC 707 Chemical Structure

CAS NO. 1687736-54-4

SGC 707 is a potent allosteric inhibitor of PRMT3 (IC50 = 50 nM) with >100-fold selectivity over other methyltransferases and other non-epigenetic targets.

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10 mg
$65.00
25 mg
$140.00
50 mg
$225.00
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Biological Activity

SGC 707 is a potent allosteric inhibitor of PRMT3 (IC50 = 50 nM) with >100-fold selectivity over other methyltransferases and other non-epigenetic targets.
Targets
PRMT3 PRMT3
31 nM53 nM(Kd)
In vitro DMSO 51 mg/mL (170.95 mM)
Water Insoluble
Ethanol Warmed: 51 mg/mL (170.95 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 33.52 mL 167.62 mL 335.23 mL
0.5 mM 6.7 mL 33.52 mL 67.05 mL
1 mM 3.35 mL 16.76 mL 33.52 mL
5 mM 0.67 mL 3.35 mL 6.7 mL

*The above data is based on the productmolecular weight 298.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15450
Actions Inhibitor
CAS No. 1687736-54-4
Formula C16H18N4O2
M. Wt 298.3
Purity >98%
Synonyms SGC707, SGC-707
SMILES C1CCN(C1)C(=O)CNC(=O)NC2=CC3=C(C=C2)C=NC=C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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