TC-E 5005 is a highly selective inhibitor of the phosphodiesterase 10A (PDE10A) enzyme, exhibiting IC50 values of 7.28 nM for PDE10A, while demonstrating significantly higher values for PDE2A, 11A, 5A, 7B, and 3A. This compound effectively inhibits adrenergic and neurogenic smooth muscle contractions in human prostate tissues, making it a valuable tool for studying PDE10A's role in smooth muscle physiology and potential therapeutic applications in urological disorders.
TC-E 5005 is a highly selective inhibitor of the phosphodiesterase 10A (PDE10A) enzyme, exhibiting IC50 values of 7.28 nM for PDE10A, while demonstrating significantly higher values for PDE2A, 11A, 5A, 7B, and 3A. This compound effectively inhibits adrenergic and neurogenic smooth muscle contractions in human prostate tissues, making it a valuable tool for studying PDE10A's role in smooth muscle physiology and potential therapeutic applications in urological disorders.
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